1.1: trichlorophosphate / 0.25 h / 25 °C
1.2: 0.5 h / 20 - 60 °C
1.3: 0.5 h
2.1: sodium; methanol / 0.5 h / |Reflux
3.1: potassium hydroxide / methanol; water / 3 h / |Reflux
View Scheme
参考文献
Sahner, J. Henning; Brengel, Christian; Storz, Michael P.; Groh, Matthias; Plaza, Alberto; Mueller, Rolf; Hartmann, Rolf W.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 21 p. 8656 - 8664