1: 80 percent / AlCl3 / CH2Cl2 / 15 h / Ambient temperature
2: 42 percent / AlCl3 / CH2Cl2 / 5 h / Heating
View Scheme
参考文献
Plattner, Jacob J.; Fung, Anthony K.L.; Smital, Jill R.; Lee, Cheuk-Man; Crowley, Steven R.; et al.
Journal of Medicinal Chemistry, 1984 , vol. 27, # 12 p. 1587 - 1596