1: 87 percent / CH2Cl2 / 4 h / Ambient temperature
2: POCl3, P2O5 / 2 h / Heating
3: H2 / PtO2 / ethanol / 10 h / 2792.6 Torr
View Scheme
参考文献
Gray, Nancy M.; Cheng, Brian K.; Mick, Stephen J.; Lair, Cecelia M.; Contreras, Patricia C.
Journal of Medicinal Chemistry, 1989 , vol. 32, # 6 p. 1242 - 1248