反应条件
1: 4-(N,N-dimethlyamino)pyridine; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride / dichloromethane / 3 h / 20 °C / Inert atmosphere 2: methanol; sodium hydroxide / tetrahydrofuran / 2 h / 20 °C View Scheme
参考文献
Tang, Yan-Bo; Lu, Dianyun; Chen, Zheng; Hu, Chun; Yang, Ying; Tian, Jin-Ying; Ye, Fei; Wu, Li; Zhang, Zhong-Yin; Xiao, Zhiyan
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 8 p. 2313 - 2318