反应条件
1: With sodium tris(acetoxy)borohydride in acetic acid; 1,2-dichloro-ethane T=20°C; 16 h; 2: With hydrogenchloride in water; acetic acid; 1,2-dichloro-ethane; acetone T=20°C; 16 h;
参考文献
AMGEN INC.; BODE, Christiane, M.; CHENG, Alan, C.; CHOQUETTE, Deborah; LEWIS, Richard, T.; POTASHMAN, Michele, H.; ROMERO, Karina; STELLWAGEN, John, C.; WHITTINGTON, Douglas, A.
Patent: WO2012/18668 A1, 2012 ;
Location in patent: Page/Page column 164 ;
WO 2012/018668 A1