1: With benzoic acid in chloroform T=-50 - -30°C; aza-Michael addition; 70 h; 2: With sodium tetrahydroborate in methanol; chloroform T=0°C; 0.5 h; Further stages. Title compound not separated from byproducts.;
参考文献
Fustero, Santos; Jimenez, Diego; Moscardo, Javier; Catalan, Silvia; Del Pozo, Carlos
Organic Letters, 2007 , vol. 9, # 25 p. 5283 - 5286