反应条件
1: With n-butyllithium; N,N,N',N,-tetramethylethylenediamine in tetrahydrofuran T=-78°C; 2 h; 2: With iodine in tetrahydrofuran T=-78°C; 1 h;
参考文献
Stoit, Axel R.; den Hartog, Arnold P.; Mons, Harry; van Schaik, Sjoerd; Barkhuijsen, Nynke; Stroomer, Cees; Coolen, Hein K.A.C.; Reinders, Jan Hendrik; Adolfs, Tiny J.P.; van der Neut, Martina; Keizer, Hiskias; Kruse, Chris G.
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 1 p. 188 - 193