1: 75 percent / NaOAc; MeNH2*HCl / methanol / 12 h / 20 °C 2: 60 percent / NaBH4 / tetrahydrofuran; methanol / 2 h / 20 °C 3: 65 percent / CsF / acetonitrile / 16 h / 70 °C View Scheme
参考文献
Ptaszek, Marcin; Bhaumik, Jayeeta; Kim, Han-Je; Taniguchi, Masahiko; Lindsey, Jonathan S.
Organic Process Research and Development, 2005 , vol. 9, # 5 p. 651 - 659