反应条件
1: With acetic acid in 1,2-dichloro-ethane T=20°C; 1 h; 2: With sodium cyanoborohydride in methanol; 1,2-dichloro-ethane Further stages.;
参考文献
Biswas, Swati; Zhang, Suhong; Fernandez, Fernando; Ghosh, Balaram; Zhen, Juan; Kuzhikandathil, Eldo; Reith, Maarten E. A.; Dutta, Aloke K.
Journal of Medicinal Chemistry, 2008 , vol. 51, # 1 p. 101 - 117