反应条件
1: 91 percent / pyridine / CH2Cl2 / 0.5 h / Ambient temperature 2: 100 percent / 1 h / 90 °C 3: 80 percent / pyridine / 72 h / 110 °C 4: 2) Amberlite IRA-410 / 1) 39 h, reflux, 2) MeOH, H2O View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 32, # 1 p. 56 - 64