6-(甲基氨基)-3-吡啶硼酸频那醇酯合成路线 (共 2 条)
反应条件
potassium acetate; dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct in N,N-dimethyl-formamide T=150°C; 0.166667 h; Microwave irradiation;
参考文献
WO2007/86800 A1, ;
Page/Page column 92-93 ;
WO 2007/086800 A1
反应条件
N-ethyl-N,N-diisopropylamine in 1,4-dioxane T=20°C; 16 h;
参考文献
WO2012/167423 A1, ;
Page/Page column 35 ;
WO 2012/167423 A1