With thionyl chloride in benzene T=15 - 20°C; 2 h;
参考文献
Reddy, M. V. Ramana; Mallireddigari, Muralidhar R.; Cosenza, Stephen C.; Pallela, Venkat R.; Iqbal, Nabisa M.; Robell, Kimberly A.; Kang, Anthony D.; Reddy, E. Premkumar Journal of Medicinal Chemistry, 2008 , vol. 51, # 1 p. 86 - 100