6-氯吡嗪-2-硼酸频那醇酯合成路线 (共 1 条)
反应条件
potassium acetate; tri-cyclo-hexyl-phosphine; tris-(dibenzylideneacetone)dipalladium(0) in 1,4-dioxane T=80°C; 18 h; Inert atmosphere;
参考文献
NOVARTIS AG; BARSANTI, Paul, A.; HU, Cheng; JIN, Xianming; NG, Simon, C.; PFISTER, Keith, B.; SENDZIK, Martin; SUTTON, James
Patent: WO2012/101064 A1, 2012 ;
Location in patent: Page/Page column 84-85 ;
WO 2012/101064 A1