1-(4-甲基-1-哌嗪)-2-[4-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯基]-乙酮合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in N,N-dimethyl-formamide T=150°C; 0.333333 h;
参考文献
NOVARTIS AG
Patent: WO2008/25512 A1, 2008 ;
Location in patent: Page/Page column 69-70 ;
WO 2008/025512 A1