反应条件
1: CH2Cl2 / 2 h / 0 °C 2: 78 percent / pyridine, 4-dimethylaminopyridine / CH2Cl2 / 3 h / 20 °C 3: 54 percent / trimethylsilyl trifluoromethanesulfonate / acetonitrile / 0.25 h / -35 °C 4: 78 percent / methylamine / ethanol / 20 °C View Scheme
参考文献
Lau; Pedersen; Nielsen
Acta chemica Scandinavica (Copenhagen, Denmark : 1989), 1991 , vol. 45, # 6 p. 616 - 620