反应条件
n-butyllithium; N,N,N',N,-tetramethylethylenediamine 1.) THF, -40 deg C, 30 min, 2.) THF, from -40 deg C to RT, overnight; Yield given. Multistep reaction;
参考文献
Harmat, Nicholas J. S.; Giorgi, Raffaello; Bonaccorsi, Fabrizio; Cerbai, Guido; Colombani, Spartaco M.; et al.
Journal of Medicinal Chemistry, 1995 , vol. 38, # 15 p. 2925 - 2937