1: dimethylformamide / 4 h / Ambient temperature 2: 45percent aq. KOH / ethanol / Heating 3: BH3*THF / 2 h / 0 °C View Scheme
参考文献
Meyer, Michael D.; Hancock, Arthur A.; Tietje, Karin; Sippy, Kevin B.; Prasad, Rajnandan; Stout, David M.; Arendsen, David L.; Donner, B. Greg; Carroll, William A.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 7 p. 1049 - 1062