反应条件
1: 78.7 percent / 15 percent NaOH / 0.75 h / Heating 2: 53.8 percent / KBr, Pb(OAc)4 / H2O; acetic acid / 30 °C 3: toluene / 3 h / Heating 4: 89 percent / PCl3 / dimethylformamide / 2 h / Ambient temperature View Scheme
参考文献
Cecchetti, Violetta; Fravolini, Arnaldo; Fringuelli, Renata; Mascellani, Giuseppe; Pagella, Piergiuseppe; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 3 p. 465 - 473