反应条件
1: p-TsOH, hexamethyldisilazane, NH3 / 120 h / 155 - 160 °C
2: 50percent aq. MeOH / 4 h / Heating
3: 100 percent / HBr / dioxane / 20 h
View Scheme
参考文献
Su, Tsann-Long; Huang, Jai-Tung; Burchenal, Joseph H.; Watanabe, Kyoichi A.; Fox, Jack J.
Journal of Medicinal Chemistry, 1986 , vol. 29, # 5 p. 709 - 715
