4-溴-2-环丙基-1H-吡咯并[2,3-b]吡啶合成路线 (共 1 条)
反应条件
1: With [14C]-Tetramethylammonium bromide; trifluoromethanesulfonic anhydride in N,N-dimethyl-formamide T=0 - 20°C; 37.1667 h; 2: With sodium hydroxide in water; N,N-dimethyl-formamide pH=11 - 12; 1 h;
参考文献
WO2009/147188 A1, ;
Page/Page column 105-106 ;
WO 2009/147188 A1