反应条件
1: 98 percent / cc. HCl / dioxane / 0.5 h / 60 °C 2: 98 percent / AlCl3 / CH2Cl2 / 24 h / 20 °C 3: 93 percent / KF / methanol / 1.) 15 h, RT; 2.) 4 h, reflux View Scheme
参考文献
Royer; Einhorn; Demerseman; et al.
European Journal of Medicinal Chemistry, 1985 , vol. 20, # 5 p. 429 - 432