反应条件
1: 86 percent / CHCl3 / Heating 2: 85 percent / dibal / toluene / -78 - 0 °C 3: 1.) KH / 1.) THF, DMF 4: 48percent aq. HF / acetonitrile / 0 °C 5: 80 percent / I2, Na2CO3 / acetonitrile / 3 h / 0 °C View Scheme
参考文献
Journal of Organic Chemistry, , vol. 51, # 12 p. 2230 - 2240