1: With sodium dithionite; triethylamine in ethanol; water
T=50°C; 1.5 h;
2: With hydrogenchloride in ethanol; water
T=60°C; 1 h; Product distribution / selectivity;
参考文献
TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION; MOUNT SINAI SCHOOL OF MEDICINE; REDDY, E., Premkumar; REDDY, M. V., Ramana
Patent: WO2012/166586 A1, 2012 ;
Location in patent: Page/Page column 74 ;
WO 2012/166586 A1