反应条件
1: 99 percent / EtONa, / ethanol / 0.08 h / Heating 2: 96 percent / SOCl2, / diethyl ether / 0.25 h / Heating 3: 62 percent / NH3, / methanol / 16 h / 100 °C 4: 86 percent / CHCl3 / 0.25 h / Heating 5: 78 percent / K2CO3, / methanol; H2O / Heating 6: ethanol / 2 h / Heating View Scheme
参考文献
Sterk; Van Der Goot; Timmerman
European Journal of Medicinal Chemistry, 1986 , vol. 21, # 4 p. 305 - 309