反应条件
benzotriazol-1-ol; triethylamine; dicyclohexyl-carbodiimide 1.) DMF, 23 deg C, 0.5 h, 2.) DMF a.) 0 deg C, 2 h, b.) 23 deg C, 15 h; Yield given. Multistep reaction;
参考文献
Lipkowski; Tam; Portoghese
Journal of Medicinal Chemistry, 1986 , vol. 29, # 7 p. 1222 - 1225