(R)-吡咯烷3-乙酸甲酯盐酸盐合成路线 (共 1 条)
反应条件
1: ((3R)-1-{[(1,1-dimethylethyl)oxy]carbonyl}-3-pyrrolidinyl)acetic acid With hydrogenchloride in 1,4-dioxane T=18 - 25°C; 20 h; 2: methanol With hydrogenchloride T=10 - 25°C;
参考文献
AstraZeneca AB
Patent: US2008/269288 A1, 2008 ;
Location in patent: Page/Page column 105 ;
US 20080269288 A1