反应条件
1: 5 N NaOH / ethanol / 3 h / Ambient temperature 2: KOH, hydrazine monohydrate, diethylene glycol / 6 h / 140 °C 3: thionyl chloride / benzene / 0.67 h / Heating 4: AlCl3 / CS2 / 4 h / Heating View Scheme
参考文献
Yoshimura; Nagai; Hibi; Kikuchi; Abe; Hida; Higashi; Yamanaka
Journal of Medicinal Chemistry, 1995 , vol. 38, # 16 p. 3163 - 3173