反应条件
1: 1.) DCC, HOBT, 4-methylmorpholine / 1.) THF, 2.) THF, DMF, 24 h 2: LiAlH4 / dioxane / 48 h / Heating View Scheme
参考文献
Breslin; Kukla; Ludovici; Mohrbacher; Ho; Miranda; Rodgers; Hitchens; Leo; Gauthier; Scott; De Clercq; Pauwels; Andries; Janssen
Journal of Medicinal Chemistry, 1995 , vol. 38, # 5 p. 771 - 793