反应条件
1: 1.) H2 / 1.) 10percent Pd/C / 2.) EtOH, Et2O
2: 95 percent / bovine trypsin, MOPS buffer (pH 8.0), CaCl2 / dimethylsulfoxide / 5 h / 25 °C
View Scheme
参考文献
Sekizaki, Haruo; Itoh, Kunihiko; Toyota, Eiko; Tanizawa, Kazutaka
Chemical and Pharmaceutical Bulletin, 1998 , vol. 46, # 5 p. 846 - 849