反应条件
4-(N,N-dimethlyamino)pyridine; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide 1 h;
参考文献
Zablocki; Rico; Garland; Rogers; Williams; Schretzman; Rao; Bovy; Tjoeng; Lindmark; Toth; Zupec; McMackins; Adams; Miyano; Markos; Milton; Paulson; Herin; et al.
Journal of Medicinal Chemistry, 1995 , vol. 38, # 13 p. 2378 - 2394