4-氟-3-(三氟甲基磺酰基)苯磺酰氯合成路线 (共 2 条)
反应条件
chlorosulfonic acid T=120°C; 18 h;
参考文献
GENENTECH, INC.; WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH
Patent: WO2008/61208 A2, 2008 ;
Location in patent: Page/Page column 30-31 ;
WO 2008/061208 A2
反应条件
ammonia in water; isopropyl alcohol T=-78°C; 2 h;
参考文献
GENENTECH, INC.; WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH
Patent: WO2008/61208 A2, 2008 ;
Location in patent: Page/Page column 30; 31 ;
WO 2008/061208 A2