1: thiophenol With sodium hydride in tetrahydrofuran
T=0 - 10°C; 1 h;
2: C17H24N2O7S in tetrahydrofuran
T=0 - 20°C; 1.5 h;
参考文献
GENENTECH, INC.; WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH
Patent: WO2008/61208 A2, 2008 ;
Location in patent: Page/Page column 31; 33 ;
WO 2008/061208 A2