反应条件
1: 4-chlorophenyl phosphorodichloridate, pyridine / 72 h / Ambient temperature 2: 1.) NH4OH, 2.) NH3 / 1.) dioxane, RT, 5 h, 2.) MeOH, RT, pressure, overnight View Scheme
参考文献
Lin; Chen; McLaren; Gao; Ghazzouli; Prusoff
Journal of Medicinal Chemistry, 1987 , vol. 30, # 2 p. 440 - 444