反应条件
1: 1.) Na / 1.) EtOH, r.t.; 2.) EtOH, 40-50 deg C, 1.5 h 2: 11 g / benzoyl peroxide, NBS / CCl4 / 8 h / Heating 3: Et3N / CH2Cl2 / 1 h / Ambient temperature View Scheme
参考文献
Ohno; Komatsu; Mizukoshi; Ichihara; Nakamura; Morishima; Sumita
Chemical and Pharmaceutical Bulletin, 1986 , vol. 34, # 4 p. 1589 - 1606