1: With magnesium in tetrahydrofuran T=20°C; 1 h; 2: With tri-isopropoxy-borane in tetrahydrofuran T=-78 - 20°C; 49 h; 3: With water T=20°C; 1 h; Further stages.;
参考文献
Contreras; Parrot; Sippl; Rival; Wermuth
Journal of Medicinal Chemistry, 2001 , vol. 44, # 17 p. 2707 - 2718