Stage #1: With dimethylsulfide borane complex in tetrahydrofuran 6 h; Heating / reflux; Stage #2: With methanol in tetrahydrofuran 2 h; Heating / reflux; Stage #3: With hydrogenchloride in water T=0°C; Product distribution / selectivity; Show Experimental Procedure
参考文献
ARENA PHARMACEUTICALS, INC. Patent: WO2008/70111 A2, 2008 ; Location in patent: Page/Page column 18-20 ;WO 2008/070111 A2