反应条件
1: 67 percent / K2CO3 / dimethylformamide / 16 h / Ambient temperature 2: 62 percent / CH2I2, iso-pentyl nitrite / tetrahydrofuran / 1 h / 85 °C 3: 66 percent / liq. NH3 / 24 h / Ambient temperature View Scheme
参考文献
Camaioni, Emidio; Costanzi, Stefano; Vittori, Sauro; Volpini, Rosaria; Klotz, Karl-Norbert; Cristalli, Gloria
Bioorganic and Medicinal Chemistry, 1998 , vol. 6, # 5 p. 523 - 533