4-氯-1-苯磺酰基-1H-吡咯并[2,3-b]吡啶-5-甲醛合成路线 （共 2 条）
反应条件
1: 4-chloro-1H-pyrrolo[2,3-b]pyridine-5-carbaldehyde With caesium carbonate in N,N-dimethyl-formamide T=20°C; 0.333333 h; 2: benzenesulfonyl chloride in N,N-dimethyl-formamide T=20°C; 2 h;
参考文献
INCYTE CORPORATION; WU, Liangxing; ZHANG, Colin; HE, Chunhong; SUN, Yaping; LU, Liang; QIAN, Ding-Quan; XU, Meizhong; ZHUO, Jincong; YAO, Wenqing
Patent: WO2014/7951 A2, 2014 ;
Location in patent: Page/Page column 216; 217 ;
反应条件
toluene-4-sulfonic acid in toluene Reflux;
参考文献
US2010/48552 A1, ;
Page/Page column 16 ;
