gsk 1292263; 5-[[[1-(3-异丙基-1,2,4-噁二唑-5-基)-4-哌啶基]甲基]氧基]-2-[4-(甲磺酰基)苯基]吡啶合成路线 (共 2 条)
反应条件
potassium carbonate in N,N-dimethyl-formamide T=80°C; 20 h;
参考文献
US2010/29650 A1, ;
Page/Page column 50 ;
反应条件
di-isopropyl azodicarboxylate; triphenylphosphine in tetrahydrofuran T=20°C; 4 h;
参考文献
US2010/29650 A1, ;
Page/Page column 82 ;