反应条件
1: 30 percent / NaH / tetrahydrofuran / 60 °C 2: 89 percent / H2, 5N HCl / Pd-C / methanol; H2O 3: 1) DIBAL-H, 2) (COCl)2, DMSO, Et3N / 1) toluene, -35 deg C -> 25 deg C, 2) CH2Cl2, -70 deg C View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 6, # 15 p. 1825 - 1830