5-碘-1H-吡唑并[3,4-c]吡啶合成路线 (共 1 条)
反应条件
1: With acetic acid in toluene 2: With potassium acetate; isopentyl nitrite in toluene T=20°C; 48 h; 3: With water; sodium hydrogencarbonate in ethyl acetate; toluene
参考文献
BAYER SCHERING PHARMA AKTIENGESELLSCHAFT
Patent: WO2008/71451 A1, 2008 ;
Location in patent: Page/Page column 53-54 ;
WO 2008/071451 A1