1-甲基-5-(2-(4-甲基哌嗪-1-基)-5-(4-甲基哌嗪-1-基磺酰基)噻吩-3-基)-3-丙基-1H-吡唑并[4,3-d]嘧啶-7(6H)-酮合成路线 (共 1 条)
反应条件
1,1'-bis-(diphenylphosphino)ferrocene; palladium diacetate; caesium carbonate in N,N-dimethyl-formamide T=120°C; 6 h;
参考文献
Chen, Gong; Wang, Huanchen; Robinson, Howard; Cai, Jiwen; Wan, Yiqian; Ke, Hengming
Biochemical Pharmacology, 2008 , vol. 75, # 9 p. 1717 - 1728