(1S)-1,5-脱水-1-C-[3-(苯并[b]噻吩-2-基甲基)-4-氟苯基]-D-山梨糖醇 2,3,4,6-四乙酸酯合成路线 (共 1 条)
反应条件
1: With methanol; water; sodium hydroxide T=25 - 49.1°C; 2: With hydrogenchloride in methanol; water T=20.2 - 60°C;
参考文献
Astellas Pharma Inc.; Kotobuki Pharmaceutical Co., Ltd.
Patent: EP2105442 A1, 2009 ;
Location in patent: Page/Page column 15 ;