1.1: 1-methyl-pyrrolidin-2-one / 16 h / 200 °C 2.1: water; lithium hydroxide hydrate / 1,4-dioxane / 1.5 h / 30 °C 2.2: 20 °C View Scheme
参考文献
ARENA PHARMACEUTICALS, INC.; JONES, Robert M.; BUZARD, Daniel J.; HAN, Sangdon; LEHMANN, Juerg; LOPEZ, Luis A.; ULLMAN, Brett; KAWASAKI, Andrew M.; THORESEN, Lars; ZHU, Xiuwen
Patent: WO2011/5290 A1, 2011 ;
WO 2011/005290 A1