(2R)-1-乙酰基-2,3-二氢-1H-吲哚-2-羧酸合成路线 (共 7 条)
反应条件
bis(1,5-cyclooctadiene)-rhodium(I) tetrafluoroborate; hydrogen; caesium carbonate; (S)-PipPhos in dichloromethane T=40°C; P=18751.9 Torr; optical yield given as percent eeenantioselective reaction;
参考文献
Mrsic, Natasa; Jerphagnon, Thomas; Minnaard, Adriaan J.; Feringa, Ben L.; de Vries, Johannes G.
Tetrahedron Asymmetry, 2010 , vol. 21, # 1 p. 7 - 10
反应条件
1: triethylamine / 100 °C 2: H2 / platinum oxide / 760 Torr View Scheme
参考文献
Stanton; Gruenfeld; Babiarz; Ackerman; Friedmann; Yuan; Macchia
Journal of Medicinal Chemistry, 1983 , vol. 26, # 9 p. 1267 - 1277
反应条件
1: H2 / platinum oxide / 760 Torr View Scheme
参考文献
Stanton; Gruenfeld; Babiarz; Ackerman; Friedmann; Yuan; Macchia
Journal of Medicinal Chemistry, 1983 , vol. 26, # 9 p. 1267 - 1277
反应条件
in N,N-dimethyl-formamide
参考文献
Ramos Tombo, Gerardo M.; Schaer, Hans-Peter; Ghisalba, Oreste
Agricultural and Biological Chemistry, 1987 , vol. 51, # 7 p. 1833 - 1838
参考文献
Stanton; Gruenfeld; Babiarz; Ackerman; Friedmann; Yuan; Macchia
Journal of Medicinal Chemistry, 1983 , vol. 26, # 9 p. 1267 - 1277
反应条件
T=24°C; Product distribution;
参考文献
Ramos Tombo, Gerardo M.; Schaer, Hans-Peter; Ghisalba, Oreste
Agricultural and Biological Chemistry, 1987 , vol. 51, # 7 p. 1833 - 1838
参考文献
Ramos Tombo, Gerardo M.; Schaer, Hans-Peter; Ghisalba, Oreste
Agricultural and Biological Chemistry, 1987 , vol. 51, # 7 p. 1833 - 1838