反应条件
1.1: N-ethyl-N,N-diisopropylamine / dichloromethane / 2 h / 20 °C
2.1: tetrabutyl ammonium fluoride / acetonitrile
3.1: sodium hydride / tetrahydrofuran / 1 h
3.2: |Darkness
4.1: hydrogenchloride / tetrahydrofuran; water / 4 h
View Scheme
参考文献
Wu, Guang-Peng; Zu, Yu-Ping; Xu, Peng-Xiang; Ren, Wei-Min; Lu, Xiao-Bing
Chemistry - An Asian Journal, 2013 , vol. 8, # 8 p. 1854 - 1862