反应条件
1: 1.) sodium hydride / 1.) THF, 40 deg C, 30 min, 2.) RT, overnight 2: 85 percent / tetrahydrofuran; diethyl ether / 2 h / -78 °C View Scheme
参考文献
Witty, David R.; Walker, Graham; Bateson, John H.; O'Hanlon, Peter J.; Cassels, Robert
Bioorganic and Medicinal Chemistry Letters, 1996 , vol. 6, # 12 p. 1375 - 1380