(1R)-5-甲氧基-1,2,3,4-四氢萘-1-基)胺合成路线 （共 2 条）
反应条件
1: 99 percent / (S,S)-N-(p-tolylsulfonyl)-1,2-diphenylethylenediamine; HCO2H; Et3N / [RuCl2(ν6-mesitylene)]2 2: diphenyl phosphorazidate; DBU / toluene 3: H2 / Pd/C / methanol View Scheme
参考文献
Abate, Carmen; Niso, Mauro; Lacivita, Enza; Mosier, Philip D.; Toscano, Annamaria; Perrone, Roberto
Journal of Medicinal Chemistry, 2011 , vol. 54, # 4 p. 1022 - 1032
反应条件
1: diphenyl phosphorazidate; DBU / toluene 2: H2 / Pd/C / methanol View Scheme
参考文献
Hattori, Kouji; Okitsu, Osamu; Tabuchi, Seiichiro; Taniguchi, Kiyoshi; Nishio, Mie; Koyama, Satoshi; Seki, Jiro; Sakane, Kazuo
Bioorganic and Medicinal Chemistry Letters, 2005 , vol. 15, # 13 p. 3279 - 3283
