反应条件
1: 42 percent / CuCl, Cu, N-ethylmorpholine / various solvent(s) / 15 h / 70 - 80 °C 2: 69 percent / NaBH4, NaOMe / methanol / Heating 3: 1.) 1,1-carbonyldiimidazole / 1.) DMF, 20 deg C, 10 min, 2.) DMF, 5 min View Scheme
参考文献
Rewcastle; Denny; Baguley
Journal of Medicinal Chemistry, 1987 , vol. 30, # 5 p. 843 - 851
