1: carbon disulfide; 4-methyl benzyl amine With sodium hydroxide T=100°C; 0.0833333 h; Microwave irradiation; 2: chloroacetic acid T=40 - 100°C; 0.0833333 h; 3: With hydrogenchloride in water T=40 - 120°C; 0.5 h;
参考文献
Nitsche, Christoph; Schreier, Verena N.; Behnam, Mira A. M.; Kumar, Anil; Bartenschlager, Ralf; Klein, Christian D.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 21 p. 8389 - 8403